New article “Structure–Activity Relationships of Potent, Targeted Covalent Inhibitors That Abolish Both the Transamidation and GTP Binding Activities of Human Tissue Transglutaminase” was recently published in the Journal of Medicinal Chemistry.
Congratulations to co-authors Abdullah Akbar and Nicole McNeil, and contributing past and present Keillors! Take a look :
http://pubs.acs.org/doi/abs/10.1021/acs.jmedchem.7b01070